
簡要描述:ELN 441958 913064-47-8ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.
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| 品牌 | absin | CAS | 913064-47-8 |
|---|---|---|---|
| 分子式 | C29H29ClN4O2 | 純度 | ≥98% |
| 分子量 | 501.02 | 貨號 | abs47027898 |
| 規(guī)格 | 10mg | 供貨周期 | 現(xiàn)貨 |
| 主要用途 | is a potent | 應(yīng)用領(lǐng)域 | 化工,生物產(chǎn)業(yè),農(nóng)林牧漁,制藥/生物制藥,綜合 |
ELN 441958 913064-47-8
| 產(chǎn)品描述 | |
| 描述 | ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. ELN-441958 is highly selective for B1 over B2 receptors, and >500/ 2000-fold selective for the B1 over _mu_/_delta_-opioid receptor. |
| 純度 | ≥98% |
| 儲存/保存方法 | Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution. |
| 基本信息 | |
| 可溶性/溶解性 | DMSO : 100 mg/mL (199.59 mM; Need ultrasonic) |
| 生物活性 | |
| 靶點(diǎn) | Bradykinin Receptor |
| 研究領(lǐng)域 | |
| 研究領(lǐng)域 | Drug DiscoverySmall Molecule DrugLead Compound Discovery |
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